SCHEMBL16585652

SCHEMBL16585652

O=C(O)c1cc(F)c(OCc2ccccc2)cc1OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.58
CTSV O60911 3/20 0.56
CTSL P07711 3/20 0.56
MRGPRX4 Q96LA9 3/20 0.54
NPC1 O15118 1/20 0.54
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
POLB P06746 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
PTGER1 P34995 3/20 0.52
MCL1 Q07820 3/20 0.50
NR4A1 P22736 1/20 0.49
NR4A2 P43354 1/20 0.49
NR4A3 Q92570 1/20 0.49
S1PR5 Q9H228 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15968165 0.91 FOLH1 (0.55) FOLH1CTSVCTSLMRGPRX4NPC1
SCHEMBL19667234 0.88 FOLH1 (0.56) FOLH1CTSVCTSLMRGPRX4NPC1
SCHEMBL31166843 0.88 MAOB (0.57) CTSVCTSLMRGPRX4NPC1L3MBTL1
SCHEMBL25298462 0.88 FOLH1 (0.55) FOLH1CTSVCTSLMRGPRX4NPC1
SCHEMBL30442197 0.88 FOLH1 (0.55) FOLH1CTSVCTSLMRGPRX4NPC1
SCHEMBL24983867 0.87 FOLH1 (0.65) FOLH1CTSVCTSLKDM4EALDH1A1
SCHEMBL30892473 0.87 FOLH1 (0.65) FOLH1CTSVCTSLKDM4EALDH1A1
SCHEMBL10089235 0.87 FOLH1 (0.69) FOLH1KDM4EALDH1A1POLBL3MBTL1
SCHEMBL20400911 0.87 FOLH1 (0.55) FOLH1CTSVCTSLMRGPRX4NPC1
SCHEMBL19679217 0.87 PTGER1 (0.55) FOLH1CTSVCTSLMRGPRX4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015040425-A1 RESORCINOL N-ARYL AMIDE COMPOUNDS, FOR USE AS PYRUVATE DEHYDROGENASE KINASE INHIBITORS VERNALIS (R&D) LIMITED (GB) 2015-03-26 WO disclosed