SCHEMBL10089235

SCHEMBL10089235

O=C(O)c1cc(OCc2ccccc2)c(C(=O)O)cc1OCc1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 2/20 0.69
ALDH1A1 P00352 2/20 0.61
KDM4E B2RXH2 1/20 0.61
POLB P06746 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
NR4A2 P43354 2/20 0.58
NR4A1 P22736 1/20 0.58
NR4A3 Q92570 1/20 0.58
MCL1 Q07820 3/20 0.57
PTGER1 P34995 3/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
SRD5A2 P31213 1/20 0.53
SGMS2 Q8NHU3 2/20 0.53
MAOB P27338 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24983867 0.96 FOLH1 (0.65) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL30892473 0.96 FOLH1 (0.65) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL23796954 0.90 ALDH1A1 (0.66) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL7273836 0.90 FOLH1 (0.61) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL26158608 0.89 FOLH1 (0.57) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL23809720 0.89 FOLH1 (0.57) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL26158612 0.89 FOLH1 (0.57) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL16416469 0.88 TSHR (0.61) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL344833 0.88 FOLH1 (0.68) FOLH1ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL383569 0.88 FOLH1 (0.60) FOLH1ALDH1A1KDM4EPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250154143-A1 PRODRUGS FOR USE IN THE TREATMENT OF TISSUE DAMAGE UCL BUSINESS LTD (GB) 2025-05-15 US disclosed
CN-115279730-B 2, 5-Or 2, 6-disubstituted hydroquinone derivatives having at least one carboxyl, sulfo or amido group, useful as medicaments OM药物公司 2025-02-14 CN disclosed
EP-4118069-B1 PARA-HYDROQUINONE DERIVATIVES AS VEGF, TNF AND/OR IL INHIBITORS FOR THE TREATMENT OF NEUROINFLAMMATORY DISEASES OM PHARMA SA (CH) 2024-10-23 EP disclosed
EP-4387619-A1 PRODRUGS FOR USE IN THE TREATMENT OF TISSUE DAMAGE UCL Business Ltd (GB) 2024-06-26 EP disclosed
US-20230150951-A1 2,5- OR 2,6-DISUBSTITUTED HYDROQUINONE DERIVATIVES WITH AT LEAST ONE CARBOXY, SULFO OR AMIDO GROUP USEFUL AS MEDICAMENTS OM PHARMA SA (CH) 2023-05-18 US disclosed
US-20230150951-A1 2,5- OR 2,6-DISUBSTITUTED HYDROQUINONE DERIVATIVES WITH AT LEAST ONE CARBOXY, SULFO OR AMIDO GROUP USEFUL AS MEDICAMENTS OM PHARMA SA (CH) 2023-05-18 US disclosed
US-20230118142-A1 AGENTS FOR USE IN THE TREATMENT OF TISSUE DAMAGE UCL BUSINESS LTD (GB) 2023-04-20 US disclosed
US-20230101069-A1 AGENTS FOR USE IN THE TREATMENT OF TISSUE DAMAGE 2 UCL BUSINESS LTD (GB) 2023-03-30 US disclosed
WO-2023021149-A1 PRODRUGS FOR USE IN THE TREATMENT OF TISSUE DAMAGE UCL BUSINESS LTD (GB) 2023-02-23 WO disclosed
EP-4118069-A1 2,5- OR 2,6-DISUBSTITUTED HYDROQUINONE DERIVATIVES WITH AT LEAST ONE CARBOXY, SULFO OR AMIDO GROUP USEFUL AS MEDICAMENTS OM Pharma SA (CH) 2023-01-18 EP disclosed
US-9102609-B2 Functionalization of organic molecules using metal-organic frameworks (MOFS) as catalysts THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-08-11 US disclosed
US-8916722-B2 Complex mixed ligand open framework materials THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-12-23 US disclosed
US-8916722-B2 Complex mixed ligand open framework materials THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-12-23 US disclosed
US-8916722-B2 Complex mixed ligand open framework materials THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-12-23 US disclosed
US-20140012039-A1 FUNCTIONALIZATION OF ORGANIC MOLECULES USING METAL-ORGANIC FRAMEWORKS (MOFS) AS CATALYSTS BASF SE (DE) 2014-01-09 US disclosed
US-20140012039-A1 FUNCTIONALIZATION OF ORGANIC MOLECULES USING METAL-ORGANIC FRAMEWORKS (MOFS) AS CATALYSTS BASF SE (DE) 2014-01-09 US disclosed
US-20120259135-A1 COMPLEX MIXED LIGAND OPEN FRAMEWORK MATERIALS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-10-11 US disclosed
US-20120259135-A1 COMPLEX MIXED LIGAND OPEN FRAMEWORK MATERIALS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-10-11 US disclosed
US-20120259135-A1 COMPLEX MIXED LIGAND OPEN FRAMEWORK MATERIALS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-10-11 US disclosed
WO-2012012495-A2 FUNCTIONALIZATION OF ORGANIC MOLECULES USING METAL-ORGANIC FRAMEWORKS (MOFS) AS CATALYSTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2012-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140012039-A1 FUNCTIONALIZATION OF ORGANIC MOLECULES USING METAL-ORGANIC FRAMEWORKS (MOFS) AS CATALYSTS POF1B, EPCAM, MGMT FOLH1 399/4885ALDH1A1 1496/4885KDM4E 1502/4885
US-20230150951-A1 2,5- OR 2,6-DISUBSTITUTED HYDROQUINONE DERIVATIVES WITH AT LEAST ONE CARBOXY, SULFO OR AMIDO GROUP USEFUL AS MEDICAMENTS HRH4, NCOA4, HRH3 FOLH1 1436/4885ALDH1A1 3025/4885KDM4E 3269/4885
US-20230101069-A1 AGENTS FOR USE IN THE TREATMENT OF TISSUE DAMAGE 2 PYGL, FGB, MMP8 FOLH1 300/4885ALDH1A1 705/4885KDM4E 4333/4885
US-20230118142-A1 AGENTS FOR USE IN THE TREATMENT OF TISSUE DAMAGE LPO, AOX1, MPO FOLH1 631/4885ALDH1A1 328/4885KDM4E 3809/4885
US-20250154143-A1 PRODRUGS FOR USE IN THE TREATMENT OF TISSUE DAMAGE CYP2B6, CBR3, CYP2A6 FOLH1 1236/4885ALDH1A1 1417/4885KDM4E 4634/4885
US-20120259135-A1 COMPLEX MIXED LIGAND OPEN FRAMEWORK MATERIALS NECTIN4, PICALM, MICA FOLH1 2158/4885ALDH1A1 4707/4885KDM4E 3935/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.