SCHEMBL16588451

SCHEMBL16588451

CC=C1CCC(=O)Nc2ccc(C)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.47
CDK5 Q00535 2/20 0.44
ROS1 P08922 1/20 0.44
ACVR1 Q04771 1/20 0.44
LRRK2 Q5S007 1/20 0.44
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MMP12 P39900 1/20 0.40
PKM P14618 3/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 1/20 0.39
RET P07949 2/20 0.39
PDGFRB P09619 1/20 0.39
PDPK1 O15530 1/20 0.39
CSNK1G1 Q9HCP0 1/20 0.39
MAPT P10636 3/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872249 0.80 CDK5 (0.49) EPHX2CDK5ROS1ACVR1LRRK2
SCHEMBL14302646 0.73 PARP10 (0.38) EPHX2CDK5ROS1ACVR1LRRK2
SCHEMBL433753 0.73 PKM (0.58) EPHX2MEN1KMT2AMMP12PKM
SCHEMBL29199433 0.73 PKM (0.58) EPHX2MEN1KMT2AMMP12PKM
SCHEMBL1184463 0.70 MMP12 (0.47) EPHX2CDK5ROS1ACVR1LRRK2
SCHEMBL29783299 0.70 MMP12 (0.47) EPHX2CDK5ROS1ACVR1LRRK2
SCHEMBL8363166 0.70 MEN1 (0.61) CDK5ROS1ACVR1LRRK2MEN1
SCHEMBL1025832 0.69 CA9 (0.62) EPHX2MMP12PKMALDH1A1
SCHEMBL29754317 0.69 CA9 (0.62) EPHX2MMP12PKMALDH1A1
SCHEMBL12653067 0.69 AHR (0.54) CDK5LRRK2MEN1KMT2ARET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493305-B1 2-AMINOINDOLE COMPOUNDS AND METHODS FOR THE TREATMENT OF MALARIA GENZYME CORP (US) 2015-03-25 EP disclosed