SCHEMBL16589999

SCHEMBL16589999

Cc1ccc2c(c1)CCC1COC(=O)N21

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 7/20 0.51
NOTUM Q6P988 3/20 0.49
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
AADAT Q8N5Z0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7340995 0.83 NOTUM (0.49) SRD5A1NOTUM
SCHEMBL7372067 0.83 NOTUM (0.49) SRD5A1NOTUM
SCHEMBL16587000 0.83 NOTUM (0.49) SRD5A1NOTUM
SCHEMBL7378144 0.83 NOTUM (0.49) SRD5A1NOTUM
SCHEMBL7366736 0.82 HTR2C (0.49) SRD5A1NOTUM
SCHEMBL8742792 0.82 HTR2C (0.49) SRD5A1NOTUM
SCHEMBL7342239 0.82 HTR2C (0.49) SRD5A1NOTUM
SCHEMBL7310227 0.79 NOTUM (0.71) SRD5A1NOTUM
SCHEMBL16586191 0.78 NOTUM (0.42) SRD5A1NOTUM
SCHEMBL19186850 0.78 NOTUM (0.45) SRD5A1NOTUMPOLBAADAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015040424-A1 TETRAHYDROISOQUINOLINE COMPOUNDS AND THEIR USE AS PYRUVATE DEHYDROGENASE KINASE INHIBITORS VERNALIS (R&D) LIMITED (GB) 2015-03-26 WO disclosed