SCHEMBL1660111

SCHEMBL1660111

CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(Cl)ccc3OC)c(F)c2)ccn1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDR2 Q16832 4/20 0.64
RAF1 P04049 10/20 0.63
ABL1 P00519 4/20 0.63
KIT P10721 4/20 0.63
PDGFRA P16234 4/20 0.63
KDR P35968 4/20 0.63
BRAF P15056 4/20 0.63
RIPK2 O43353 3/20 0.63
EPHX2 P34913 3/20 0.63
RET P07949 3/20 0.63
FGFR1 P11362 3/20 0.63
FLT1 P17948 3/20 0.63
EPHA1 P21709 3/20 0.63
TTK P33981 3/20 0.63
FLT4 P35916 3/20 0.63
FLT3 P36888 3/20 0.63
CLK1 P49759 3/20 0.63
LIMK1 P53667 3/20 0.63
CDK17 Q00537 3/20 0.63
TEK Q02763 3/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1660178 0.91 RAF1 (0.68) DDR2RAF1ABL1KITPDGFRA
SCHEMBL1659561 0.90 RAF1 (0.61) DDR2RAF1ABL1KITPDGFRA
SCHEMBL1662382 0.90 DDR2 (0.51) DDR2RAF1ABL1KITPDGFRA
SCHEMBL1661876 0.90 MAPK14 (0.71) DDR2RAF1ABL1KITPDGFRA
SCHEMBL1660353 0.89 RAF1 (0.63) DDR2RAF1ABL1KITPDGFRA
SCHEMBL1662323 0.89 RAF1 (0.75) DDR2RAF1ABL1KITPDGFRA
SCHEMBL14911164 0.87 ABL1 (0.73) DDR2RAF1ABL1KITPDGFRA
SCHEMBL19888727 0.87 RAF1 (0.75) DDR2RAF1ABL1KITPDGFRA
SCHEMBL15574169 0.84 DDR2 (0.82) DDR2RAF1ABL1KITPDGFRA
SCHEMBL15575322 0.83 KMT2A (0.62) DDR2RAF1ABL1KITPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046991-A2 CERTAIN SUBSTITUTED UREAS AS MODULATORS OF KINASE ACTIVITY GILEAD CONNECTICUT, INC. (US) 2011-04-21 WO claimed
WO-2011046991-A2 CERTAIN SUBSTITUTED UREAS AS MODULATORS OF KINASE ACTIVITY GILEAD CONNECTICUT, INC. (US) 2011-04-21 WO disclosed