SCHEMBL16608985

SCHEMBL16608985

COC(=O)c1ccc(Nc2ccccc2)cc1F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.55
ALOX15 P16050 1/20 0.55
KMT2A Q03164 9/20 0.49
MEN1 O00255 8/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPK13 O15264 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
HPGD P15428 1/20 0.45
ALOX12 P18054 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
ALDH1A1 P00352 3/20 0.45
HSP90AA1 P07900 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9647595 0.85 MAPT (0.60) MAPTALOX15KMT2AMEN1LMNA
SCHEMBL16608984 0.83 MEN1 (0.54) MAPTALOX15KMT2AMEN1NPC1
SCHEMBL26436184 0.83 MAPT (0.57) MAPTALOX15KMT2AMEN1NPC1
SCHEMBL4218044 0.82 MAPT (0.61) MAPTALOX15KMT2AMEN1AKR1C3
SCHEMBL16645313 0.81 HDAC1 (0.57) MAPTALOX15KMT2AMEN1RAB9A
SCHEMBL28901159 0.81 MAPT (0.55) MAPTALOX15KMT2AMEN1LMNA
SCHEMBL28901163 0.81 MAPK13 (0.63) MAPTALOX15KMT2AMEN1NPC1
SCHEMBL29116429 0.81 SMN1; SMN2 (0.51) MAPTKMT2AMEN1NPC1RAB9A
SCHEMBL4238913 0.81 RAB9A (0.66) MAPTKMT2AMEN1NPC1RAB9A
SCHEMBL29151820 0.81 MAPT (0.51) MAPTALOX15KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115073468-B Preparation and application of imidazopyrazines BTK inhibitor 药雅科技(上海)有限公司 2023-12-22 CN disclosed
CN-115073468-A Preparation and application of imidazopyrazine BTK inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed
WO-2015048306-A1 NOVEL AGENTS TARGETING CYP51 THE SCRIPPS RESEARCH INSTITUTE (US) 2015-04-02 WO disclosed