SCHEMBL16645313

SCHEMBL16645313

COC(=O)c1ccc(Nc2ccccc2N)cc1F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.57
MAPK14 Q16539 10/20 0.55
MAPK13 O15264 8/20 0.55
MAPK12 P53778 8/20 0.55
MAPK11 Q15759 8/20 0.55
HSD17B10 Q99714 4/20 0.50
ALDH1A1 P00352 3/20 0.50
CFTR P13569 2/20 0.50
MAPT P10636 5/20 0.49
ALOX15 P16050 2/20 0.49
GAA P10253 4/20 0.48
KDM4E B2RXH2 4/20 0.48
TDP1 Q9NUW8 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
THRB P10828 1/20 0.48
HTT P42858 1/20 0.48
RECQL P46063 1/20 0.48
MMP14 P50281 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3845029 0.87 MAPK14 (0.54) HDAC1MAPK14MAPK13MAPK12MAPK11
SCHEMBL7200687 0.83 MAPK14 (0.76) HDAC1MAPK14MAPK13MAPK12MAPK11
SCHEMBL21463821 0.82 MAPK14 (0.64) MAPK14MAPK13MAPK12MAPK11HSD17B10
SCHEMBL30615339 0.82 MAPK14 (0.64) MAPK14MAPK13MAPK12MAPK11HSD17B10
SCHEMBL16608985 0.81 MAPT (0.55) MAPK14MAPK13MAPK12MAPK11ALDH1A1
SCHEMBL27482085 0.81 MAPK13 (0.72) HDAC1MAPK14MAPK13MAPK12MAPK11
SCHEMBL6812866 0.81 MAPK14 (0.81) HDAC1MAPK14MAPK13MAPK12MAPK11
SCHEMBL22101263 0.77 RAB9A (0.47) ALDH1A1MAPTALOX15KDM4EMEN1
SCHEMBL3499186 0.77 SIRT2 (0.68) HDAC1MAPK14MAPK13MAPK12MAPK11
SCHEMBL2314122 0.76 HSD17B10 (0.68) MAPK14MAPK13MAPK12MAPK11HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed