SCHEMBL16610338

SCHEMBL16610338

O=Cc1cc(Br)c(Br)c(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
ALDH1A3 P47895 2/20 0.33
ALDH1A1 P00352 2/20 0.32
GRIA1 P42261 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA3 P42263 1/20 0.31
GRIA4 P48058 1/20 0.31
ALDH3A1 P30838 1/20 0.31
NOTUM Q6P988 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3309062 0.82 KIF11 (0.39) KIF11ALDH1A3ALDH1A1
SCHEMBL27977385 0.81 KIF11 (0.38) KIF11ALDH1A3ALDH1A1GRIA1GRIA2
SCHEMBL7814448 0.78 APEX1 (0.45) ALDH1A3ALDH1A1ALDH3A1
SCHEMBL6515872 0.77 KIF11 (0.43) KIF11ALDH1A1GRIA1GRIA2GRIA3
SCHEMBL6856881 0.76 KIF11 (0.46) KIF11ALDH1A1GRIA1GRIA2GRIA3
SCHEMBL7147339 0.76 KIF11 (0.51) KIF11ALDH1A3ALDH1A1GRIA1GRIA2
SCHEMBL5546389 0.76 KIF11 (0.47) KIF11ALDH1A3ALDH1A1ALDH3A1NOTUM
SCHEMBL29417742 0.76 KIF11 (0.51) KIF11ALDH1A3ALDH1A1GRIA1GRIA2
SCHEMBL16610339 0.75 EIF2AK2 (0.47) ALDH1A1AKR1C3AKR1C2
SCHEMBL816357 0.74 KIF11 (0.44) KIF11GRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed