SCHEMBL16610339

SCHEMBL16610339

O=C(O)/C=C/c1cc(Br)c(Br)c(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF2AK2 P19525 1/20 0.47
CSNK2A2 P19784 1/20 0.47
CSNK2B P67870 1/20 0.47
CSNK2A1 P68400 1/20 0.47
KDM4E B2RXH2 4/20 0.47
GAA P10253 2/20 0.47
AKR1C3 P42330 2/20 0.45
AKR1C2 P52895 1/20 0.45
THRB P10828 2/20 0.39
THRA P10827 1/20 0.39
HDAC3 O15379 3/20 0.39
HDAC1 Q13547 3/20 0.39
HDAC2 Q92769 3/20 0.39
HDAC10 Q969S8 3/20 0.39
HDAC11 Q96DB2 3/20 0.39
HDAC8 Q9BY41 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC5 Q9UQL6 3/20 0.39
HDAC4 P56524 2/20 0.39
HDAC7 Q8WUI4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16241694 0.81 AKR1C3 (0.57) CSNK2A2CSNK2BCSNK2A1KDM4EGAA
SCHEMBL16241693 0.81 AKR1C3 (0.57) CSNK2A2CSNK2BCSNK2A1KDM4EGAA
SCHEMBL16610454 0.77 ITGB2 (0.42) KDM4EGAATHRBTHRAHDAC3
SCHEMBL16610337 0.76 TRPV1 (0.46) KDM4EHDAC3HDAC1HDAC2HDAC10
SCHEMBL16610338 0.75 KIF11 (0.40) AKR1C3AKR1C2ALDH1A1
SCHEMBL16048499 0.74 KDM4E (0.61) CSNK2A2CSNK2BCSNK2A1KDM4EGAA
SCHEMBL16048498 0.74 KDM4E (0.61) CSNK2A2CSNK2BCSNK2A1KDM4EGAA
SCHEMBL3917700 0.73 KDM4E (0.70) EIF2AK2CSNK2A2CSNK2BCSNK2A1KDM4E
SCHEMBL3917704 0.73 KDM4E (0.70) EIF2AK2CSNK2A2CSNK2BCSNK2A1KDM4E
SCHEMBL692664 0.72 KDM4E (0.50) CSNK2A2CSNK2BCSNK2A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed