SCHEMBL16612449

SCHEMBL16612449

CN(C(=O)O)C1CCN(c2ccncc2F)CC1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 13/20 0.45
NPY5R Q15761 2/20 0.43
CACNA2D1 P54289 1/20 0.41
ROCK2 O75116 1/20 0.40
PRKG1 Q13976 1/20 0.40
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15771417 0.85 MAPT (0.46) CYP46A1NPY5RCA12CA1CA2
SCHEMBL16622465 0.81 SIGMAR1 (0.47) CYP46A1NPY5RCACNA2D1CA12CA1
SCHEMBL785159 0.78 F10 (0.51) NPY5R
SCHEMBL13622696 0.76 FFAR4 (0.48) CA12CA1CA2CA9
SCHEMBL20755270 0.76 GAA (0.46) ROCK2PRKG1CDK8CA12CA1
SCHEMBL25246297 0.75 USP30 (0.44) CYP46A1
SCHEMBL19555543 0.75 CHRM4 (0.54) CYP46A1CDK8
SCHEMBL785732 0.74 GPR119 (0.52) CYP46A1CCNCCDK8
SCHEMBL784900 0.73 MCHR1 (0.46) CCNCCDK8
SCHEMBL15718658 0.72 FFAR1 (0.51) NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857388-A1 Azoles containing sulfone Grünenthal GmbH (DE) 2015-04-08 EP disclosed