SCHEMBL16612528

SCHEMBL16612528

CC1(C)CC(=O)CCC1NCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 5/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
APEX1 P27695 1/20 0.40
OPRM1 P35372 2/20 0.40
OPRL1 P41146 2/20 0.40
TSHR P16473 1/20 0.39
IDO1 P14902 1/20 0.39
ALDH1A1 P00352 1/20 0.38
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
BACE1 P56817 1/20 0.37
FABP6 P51161 1/20 0.36
RAB9A P51151 1/20 0.36
KDM1A O60341 1/20 0.36
MAOA P21397 1/20 0.36
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
SLC1A2 P43004 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29872456 0.83 MEN1 (0.45) MEN1KMT2ATSHRALDH1A1RAB9A
SCHEMBL785570 0.75 ALDH1A1 (0.50) MEN1KMT2ATSHRALDH1A1ACHE
SCHEMBL571765 0.73 GRIN2B (0.71) GRIN2BMEN1KMT2AOPRM1OPRL1
SCHEMBL31682505 0.72 GRIN2B (0.44) GRIN2BMEN1KMT2AOPRM1OPRL1
SCHEMBL16612591 0.72 FUCA1 (0.42) GRIN2BMEN1KMT2AOPRM1OPRL1
SCHEMBL4371247 0.72 GRIN2B (0.41) GRIN2BMEN1KMT2AOPRM1OPRL1
SCHEMBL6098218 0.72 PSEN1 (0.45) OPRM1OPRL1IDO1ALDH1A1
SCHEMBL12061489 0.71 CARM1 (0.45) GRIN2BMEN1KMT2AOPRM1OPRL1
SCHEMBL7723868 0.70 GRIN2B (0.66) GRIN2BMEN1KMT2AOPRM1OPRL1
SCHEMBL12699061 0.70 GRIN2B (0.41) GRIN2BMEN1KMT2AOPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857388-A1 Azoles containing sulfone Grünenthal GmbH (DE) 2015-04-08 EP disclosed
EP-2857388-A1 Azoles containing sulfone Grünenthal GmbH (DE) 2015-04-08 EP disclosed