SCHEMBL16612707

SCHEMBL16612707

NC(=O)c1n[c]cn1CCNc1nc2ccccc2o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.39
RAB9A P51151 9/20 0.39
GAA P10253 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
CSNK1D P48730 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
SCD O00767 1/20 0.37
HCRTR2 O43614 3/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
ABL1 P00519 1/20 0.36
NTRK1 P04629 1/20 0.36
LCK P06239 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612797 0.78 HCRTR2 (0.40) NPC1RAB9AGAASMN1; SMN2TP53
SCHEMBL12479212 0.76 FDPS (0.45) HCRTR2PCSK9
SCHEMBL2970656 0.71 HDAC3 (0.42) MEN1KMT2AALDH1A1KDM4ETDP1
SCHEMBL4686905 0.70 NPC1 (0.51) NPC1RAB9AGAASMN1; SMN2TP53
SCHEMBL1990188 0.68 KDM4E (0.53) NPC1RAB9AGAASMN1; SMN2TP53
SCHEMBL4686908 0.68 NPC1 (0.55) NPC1RAB9AGAASMN1; SMN2TP53
SCHEMBL1985103 0.68 NPC1 (0.52) NPC1RAB9AGAASMN1; SMN2TP53
SCHEMBL2972716 0.68 CYP1A2 (0.45) GAASMN1; SMN2ALDH1A1KDM4ETDP1
SCHEMBL25057028 0.67 NPC1 (0.50) NPC1RAB9AGAASMN1; SMN2TP53
SCHEMBL2819999 0.67 PIM3 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed