SCHEMBL16612797

SCHEMBL16612797

NC(=O)c1[c]cn(CCNc2nc3ccccc3o2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 3/20 0.40
NPC1 O15118 11/20 0.39
RAB9A P51151 11/20 0.39
GAA P10253 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
CSNK1D P48730 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
KDM4E B2RXH2 1/20 0.37
SCD O00767 1/20 0.37
TNF P01375 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
PKM P14618 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HPGD P15428 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12479961 0.85 HCRTR2 (0.43) HCRTR2GAATP53MEN1KMT2A
SCHEMBL16612707 0.78 NPC1 (0.39) HCRTR2NPC1RAB9AGAASMN1; SMN2
SCHEMBL16612601 0.78 DDAH1 (0.50) NPC1RAB9AGAASMN1; SMN2ALDH1A1
SCHEMBL16612923 0.78 LTA4H (0.43) HCRTR2NPC1RAB9ASMN1; SMN2TP53
SCHEMBL16612710 0.77 KDM4E (0.49) HCRTR2NPC1RAB9AGAASMN1; SMN2
SCHEMBL16612683 0.76 FDPS (0.45) HCRTR2
SCHEMBL4686905 0.70 NPC1 (0.51) NPC1RAB9AGAASMN1; SMN2TP53
SCHEMBL12479677 0.70 HCRTR2 (0.47) HCRTR2NPC1RAB9AGAASMN1; SMN2
SCHEMBL16612915 0.70 APAF1 (0.45) SMN1; SMN2TP53ALDH1A1KMT2ATDP1
SCHEMBL16612739 0.69 TDP1 (0.54) NPC1SMN1; SMN2ALDH1A1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed