SCHEMBL16612931

SCHEMBL16612931

CC1CCCN1C1CCN(c2ccc3c(c2)CCN(c2ccc(F)cn2)C3)C1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 17/20 0.46
KCNH2 Q12809 6/20 0.46
ADRA1A P35348 1/20 0.40
CHIA Q9BZP6 1/20 0.40
CYP3A4 P08684 1/20 0.39
GPR119 Q8TDV5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14736897 1.00 HRH3 (0.46) HRH3KCNH2ADRA1ACHIACYP3A4
SCHEMBL12181943 0.89 HRH3 (0.46) HRH3KCNH2CYP3A4GPR119
SCHEMBL12181944 0.88 GPR119 (0.40) HRH3KCNH2GPR119
SCHEMBL12181957 0.84 GPR119 (0.43) HRH3ADRA1ACHIAGPR119
SCHEMBL16612501 0.84 HRH3 (0.47) HRH3KCNH2CYP3A4
SCHEMBL2596398 0.84 HRH3 (0.47) HRH3KCNH2CYP3A4
SCHEMBL12181996 0.83 GPR119 (0.43) HRH3KCNH2CYP3A4GPR119
SCHEMBL12182151 0.82 GRIN2D (0.51) HRH3KCNH2CHIACYP3A4
SCHEMBL2596385 0.82 HRH3 (0.43) HRH3KCNH2CYP3A4
SCHEMBL12182110 0.82 HRH3 (0.44) HRH3KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569305-B1 SUBSTITUTED N-HETEROARYL TETRAHYDRO-ISOQUINOLINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2015-04-08 EP claimed