SCHEMBL1661650

SCHEMBL1661650

O=C(O)c1nc2ccc(C3(c4ccccc4)C=C3)nc2s1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.42
S1PR3 Q99500 5/20 0.35
NPC1 O15118 1/20 0.34
PKM P14618 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
S1PR5 Q9H228 1/20 0.34
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661648 0.82 S1PR1 (0.59) S1PR1S1PR3S1PR5
SCHEMBL31229583 0.72 MAPT (0.35) NPC1PKMNFKB1RAB9ANFKB2
SCHEMBL1661618 0.71 S1PR1 (0.58) S1PR1S1PR3NPC1RAB9ASMN1; SMN2
SCHEMBL1661173 0.71 ALDH1A1 (0.34) S1PR1
SCHEMBL31515643 0.71 MGAM (0.43) RAB9AMEN1MAPTKMT2ANPSR1
SCHEMBL19899747 0.69 HRH3 (0.37) SMN1; SMN2MEN1MAPTKMT2ANPSR1
SCHEMBL31493447 0.69 HRH3 (0.37) SMN1; SMN2MEN1MAPTKMT2ANPSR1
SCHEMBL1661196 0.69 S1PR1 (0.39) S1PR1S1PR3NPC1RAB9ASMN1; SMN2
SCHEMBL1661615 0.69 MAOB (0.40) S1PR1S1PR3S1PR5
SCHEMBL1661178 0.68 S1PR1 (0.56) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2306994-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF Amgen, Inc (US) 2011-04-13 EP disclosed
WO-2009154775-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF AMGEN INC. (US) 2009-12-23 WO disclosed