SCHEMBL16616897

SCHEMBL16616897

COc1cc(C=CC(=O)c2cccnc2Nc2ccc([N+](=O)[O-])cc2)cc(OC)c1OC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 3/20 0.60
MAPT P10636 4/20 0.55
ALDH1A1 P00352 4/20 0.55
LMNA P02545 2/20 0.55
HTT P42858 1/20 0.55
PTGS2 P35354 1/20 0.51
CYP1A1 P04798 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP1B1 Q16678 2/20 0.48
AMY1A P0DUB6 1/20 0.46
CYP2C8 P10632 1/20 0.46
CYP2D6 P10635 1/20 0.46
RAB9A P51151 2/20 0.46
NTSR1 P30989 1/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ABCB1 P08183 1/20 0.45
DBH P09172 1/20 0.45
NPC1 O15118 1/20 0.45
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16616893 1.00 KRAS (0.60) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616507 0.91 CYP19A1 (0.52) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616510 0.91 CYP19A1 (0.52) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616414 0.90 KRAS (0.48) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616413 0.90 KRAS (0.48) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616746 0.88 RAB9A (0.49) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616744 0.88 RAB9A (0.49) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616365 0.88 ALDH1A1 (0.57) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616410 0.88 ALDH1A1 (0.58) KRASMAPTALDH1A1LMNAHTT
SCHEMBL16616404 0.88 ALDH1A1 (0.58) KRASMAPTALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9006451-B1 2-anilinonicotinyl based chalcones useful as potential anticancer agents and process for preparation thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2015-04-14 US disclosed
US-20150099888-A1 2-Anilinonicotinyl Based Chalcones Useful As Potential Anticancer Agents and Process for Preparation Thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2015-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150099888-A1 2-Anilinonicotinyl Based Chalcones Useful As Potential Anticancer Agents and Process for Preparation Thereof HCCS, WEE2, WEE1 KRAS 1079/4885MAPT 2681/4885ALDH1A1 1497/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.