SCHEMBL16619338

SCHEMBL16619338

COc1cc2c(N[C@@H](C)c3ccccc3)c([N+](=O)[O-])cnc2cc1-c1c(C)noc1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.55
CYP3A4 P08684 12/20 0.55
CYP2C9 P11712 12/20 0.55
BRD2 P25440 11/20 0.55
BRD3 Q15059 11/20 0.55
BRDT Q58F21 2/20 0.51
CYP2C19 P33261 2/20 0.48
PDE4B Q07343 2/20 0.48
CACNA1A O00555 1/20 0.48
CHRNA1 P02708 1/20 0.48
CYP2D6 P10635 1/20 0.48
CCL2 P13500 1/20 0.48
KCNA5 P22460 1/20 0.48
TACR1 P25103 1/20 0.48
MAOB P27338 1/20 0.48
AVPR1A P37288 1/20 0.48
KCNH2 Q12809 1/20 0.48
SCN5A Q14524 1/20 0.48
CREBBP Q92793 1/20 0.48
KCNH3 Q9ULD8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11909203 1.00 BRD4 (0.55) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL16618802 0.90 CYP3A4 (0.47) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL1907697 0.90 BRD4 (0.57) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL18249949 0.87 BRD4 (0.48) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL13731782 0.87 BRD4 (0.48) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL16619839 0.87 BRD4 (0.59) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL11909184 0.87 BRD4 (0.59) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL16618930 0.86 BRD4 (0.44) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL16618838 0.86 CYP3A4 (0.55) BRD4CYP3A4CYP2C9BRD2BRD3
SCHEMBL16619069 0.85 CYP3A4 (0.54) BRD4CYP3A4CYP2C9BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049629-A1 IMIDAZOQUINOLINE COMPOUNDS AS BROMODOMAIN INHIBITORS Piramal Enterprises Limited (IN) 2015-04-09 WO disclosed