SCHEMBL16618802

SCHEMBL16618802

COC(=O)COc1cc2c(N[C@H](C)c3ccccc3)c([N+](=O)[O-])cnc2cc1-c1c(C)noc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 13/20 0.47
CYP2C9 P11712 12/20 0.47
BRD4 O60885 14/20 0.46
BRD2 P25440 9/20 0.45
BRD3 Q15059 9/20 0.45
BRDT Q58F21 2/20 0.44
PDE4B Q07343 2/20 0.41
CYP2C19 P33261 1/20 0.41
TRIM24 O15164 1/20 0.40
BRD1 O95696 1/20 0.40
CHRNA1 P02708 1/20 0.40
CHRM2 P08172 1/20 0.40
CCL2 P13500 1/20 0.40
DRD2 P14416 1/20 0.40
TAF1 P21675 1/20 0.40
DRD4 P21917 1/20 0.40
ACHE P22303 1/20 0.40
SLC6A2 P23975 1/20 0.40
MAOB P27338 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16618930 0.91 BRD4 (0.44) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL11909203 0.90 BRD4 (0.55) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619338 0.90 BRD4 (0.55) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619406 0.82 BRD4 (0.44) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619386 0.82 BRD4 (0.43) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619324 0.80 CYP3A4 (0.48) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL1907697 0.80 BRD4 (0.57) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619529 0.79 LMNA (0.55) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL16619532 0.79 LMNA (0.55) CYP3A4CYP2C9BRD4BRD2BRD3
SCHEMBL17967387 0.79 BRD4 (0.49) CYP3A4CYP2C9BRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015049629-A1 IMIDAZOQUINOLINE COMPOUNDS AS BROMODOMAIN INHIBITORS Piramal Enterprises Limited (IN) 2015-04-09 WO disclosed