SCHEMBL16620824

SCHEMBL16620824

O=C(Nc1ccc(Oc2cccc3cccnc23)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.65
BRAF P15056 9/20 0.64
CDK8 P49336 5/20 0.59
RAF1 P04049 5/20 0.59
MEN1 O00255 1/20 0.57
PLK4 O00444 1/20 0.57
CIT O14578 1/20 0.57
AURKA O14965 1/20 0.57
MUSK O15146 1/20 0.57
EPHB6 O15197 1/20 0.57
MAPK13 O15264 1/20 0.57
MLNR O43193 1/20 0.57
MAP3K7 O43318 1/20 0.57
RIPK2 O43353 1/20 0.57
DYRK3 O43781 1/20 0.57
PDE6D O43924 1/20 0.57
NR1I2 O75469 1/20 0.57
STK10 O94804 1/20 0.57
CDK14 O94921 1/20 0.57
ABCB11 O95342 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16621015 0.88 KDR (0.70) KDRBRAFCDK8RAF1MEN1
SCHEMBL16621064 0.84 BRAF (0.55) KDRBRAFCDK8RAF1PLK4
SCHEMBL29664907 0.83 RAF1 (0.68) KDRBRAFCDK8RAF1MEN1
SCHEMBL1412957 0.83 RAF1 (0.68) KDRBRAFCDK8RAF1MEN1
SCHEMBL16621229 0.82 NPC1 (0.57) KDRBRAFRAF1MAPK1EPHX2
SCHEMBL2579421 0.81 KDR (0.74) KDRBRAFCDK8RAF1RIPK1
SCHEMBL5899313 0.80 BRAF (0.57) KDRBRAFCDK8RAF1MEN1
SCHEMBL2577878 0.79 KDR (0.70) KDRBRAFCDK8RAF1MEN1
SCHEMBL936533 0.79 RAF1 (0.73) KDRBRAFCDK8RAF1MEN1
SCHEMBL30462521 0.79 RAF1 (0.73) KDRBRAFCDK8RAF1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051149-A1 SORAFENIB ANALOGS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-04-09 WO disclosed
WO-2015051149-A1 SORAFENIB ANALOGS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-04-09 WO disclosed