SCHEMBL16620989

SCHEMBL16620989

O=C(Nc1ccc(Oc2cccnc2)cc1)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.69
BRAF P15056 3/20 0.64
MAPK14 Q16539 3/20 0.64
TNNI3K Q59H18 3/20 0.64
EGFR P00533 1/20 0.60
FGFR1 P11362 1/20 0.60
CDK8 P49336 4/20 0.58
CDK7 P50613 1/20 0.58
CDK6 Q00534 1/20 0.58
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
GAA P10253 1/20 0.55
HPGD P15428 1/20 0.55
FLT3 P36888 1/20 0.54
EPHX2 P34913 1/20 0.54
RAF1 P04049 2/20 0.54
TRPV1 Q8NER1 1/20 0.53
TNF P01375 1/20 0.53
NOD1 Q9Y239 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL939205 0.86 KDR (0.79) KDRBRAFMAPK14TNNI3KEGFR
SCHEMBL11029731 0.83 TLR8 (0.62) KDRBRAFMAPK14TNNI3KCDK8
SCHEMBL16628062 0.82 RAF1 (0.76) KDRBRAFMAPK14TNNI3KEGFR
SCHEMBL11002296 0.80 TLR8 (0.62) KDRBRAFMAPK14TNNI3KCDK8
SCHEMBL16628083 0.80 KDR (0.58) KDRBRAFMAPK14TNNI3KCDK8
SCHEMBL16621239 0.79 EPHX2 (0.69) KDRBRAFMAPK14TNNI3KCDK8
SCHEMBL14527419 0.79 RAB9A (0.55) MAPK14NPC1RAB9AGAAHPGD
SCHEMBL3177619 0.78 KDR (1.00) KDRBRAFMAPK14TNNI3KCDK8
SCHEMBL938662 0.78 KDR (0.69) KDRBRAFMAPK14TNNI3KEGFR
SCHEMBL16620514 0.78 KDR (0.56) KDRBRAFMAPK14TNNI3KCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051149-A1 SORAFENIB ANALOGS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-04-09 WO disclosed
WO-2015051149-A1 SORAFENIB ANALOGS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-04-09 WO disclosed