SCHEMBL16621908

SCHEMBL16621908

O=C(c1csc(-c2ccccn2)n1)N1CCN(c2cc(Cl)ncn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
HTR2C P28335 3/20 0.44
TSHR P16473 2/20 0.44
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TACR3 P29371 1/20 0.43
HPGD P15428 2/20 0.43
SMO Q99835 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
HSD17B10 Q99714 5/20 0.43
KDM4E B2RXH2 4/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SLC6A7 Q99884 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623163 0.84 ALDH1A1 (0.41) ALDH1A1HTR2CTSHRMEN1POLB
SCHEMBL624219 0.84 ALDH1A1 (0.42) ALDH1A1HTR2CTSHRMEN1POLB
SCHEMBL623490 0.82 ALDH1A1 (0.39) ALDH1A1HTR2CTSHRMEN1POLB
SCHEMBL624238 0.82 L3MBTL1 (0.44) ALDH1A1HTR2CTSHRMEN1KMT2A
SCHEMBL623132 0.72 PTGDR2 (0.42) ALDH1A1HTR2CHPGDTLR7KDM4E
SCHEMBL622745 0.69 IRAK4 (0.47) TLR7
SCHEMBL623783 0.69 PTGDR2 (0.43) HTR2CTLR7
SCHEMBL624123 0.69 PTGDR2 (0.43) ALDH1A1HTR2CL3MBTL1TLR7SLC6A7
SCHEMBL2550713 0.68 PDE10A (0.57) ALDH1A1KMT2AL3MBTL1TLR7HSD17B10
SCHEMBL17953075 0.68 PTGDR2 (0.54) HTR2CTLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8999974-B2 Acyl piperazine derivatives as TTX-S blockers RAQUALIA PHARMA INC. (JP) 2015-04-07 US disclosed
US-8999974-B2 Acyl piperazine derivatives as TTX-S blockers RAQUALIA PHARMA INC. (JP) 2015-04-07 US disclosed