SCHEMBL16623281

SCHEMBL16623281

COc1ccc2oc(CN=O)cc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.51
CA2 P00918 3/20 0.50
KDM4E B2RXH2 5/20 0.48
ALDH1A1 P00352 5/20 0.48
HPGD P15428 4/20 0.48
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA9 Q16790 2/20 0.48
CA3 P07451 1/20 0.48
CA6 P23280 1/20 0.48
CA5A P35218 1/20 0.48
CA7 P43166 1/20 0.48
CA14 Q9ULX7 1/20 0.48
CA5B Q9Y2D0 1/20 0.48
PDE3B Q13370 1/20 0.48
PDE3A Q14432 1/20 0.48
GPR55 Q9Y2T6 1/20 0.47
MAOB P27338 3/20 0.46
APP P05067 1/20 0.46
NPC1 O15118 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1287525 0.80 CYP2A6 (0.53) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL13076441 0.79 CYP2A6 (0.51) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL1450985 0.79 CYP2A6 (0.51) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL6871528 0.79 CA2 (0.54) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL119314 0.79 CYP2A6 (0.51) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL119001 0.79 CYP2A6 (0.51) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL1287554 0.78 CYP2A6 (0.51) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL3902827 0.77 KDM4E (0.57) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL28093784 0.76 CYP2A6 (0.49) CYP2A6CA2KDM4EALDH1A1HPGD
SCHEMBL16623287 0.75 SLC22A12 (0.40) CYP2A6KDM4EALDH1A1HPGDMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857018-A1 Treatment or prophylaxis of proliferative conditions University Court of The University of Dundee (GB) 2015-04-08 EP disclosed