SCHEMBL1662329

SCHEMBL1662329

Cc1nc2ccc(C=Cc3ccccc3)nc2s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.50
RAB9A P51151 7/20 0.50
ALDH1A1 P00352 6/20 0.50
GRM4 Q14833 5/20 0.50
NPC1 O15118 4/20 0.50
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
SMN1; SMN2 Q16637 4/20 0.50
HPGD P15428 3/20 0.50
PKM P14618 2/20 0.50
LMNA P02545 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
NFKB1 P19838 2/20 0.50
GRM5 P41594 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661528 0.76 KDM4E (0.46) KDM4ERAB9AALDH1A1GRM4NPC1
SCHEMBL1661513 0.76 GRM4 (0.46) KDM4ERAB9AALDH1A1GRM4NPC1
SCHEMBL9256292 0.75 CCR1 (0.41) KDM4ERAB9AALDH1A1NPC1MEN1
SCHEMBL31003229 0.75 CCR1 (0.41) KDM4ERAB9AALDH1A1NPC1MEN1
SCHEMBL1661557 0.75 NPC1 (0.43) KDM4ERAB9AALDH1A1GRM4NPC1
SCHEMBL9169404 0.72 KDM4E (0.70) KDM4ERAB9AALDH1A1GRM4NPC1
SCHEMBL29021923 0.70 KDM4E (0.72) KDM4ERAB9AALDH1A1GRM4NPC1
SCHEMBL6312457 0.68 GRM5 (0.69) KDM4ERAB9AALDH1A1GRM4NPC1
SCHEMBL6312461 0.68 GRM5 (0.69) KDM4ERAB9AALDH1A1GRM4NPC1
SCHEMBL805088 0.68 SMN1; SMN2 (0.42) KDM4ERAB9AALDH1A1NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2306994-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF Amgen, Inc (US) 2011-04-13 EP disclosed
WO-2009154775-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF AMGEN INC. (US) 2009-12-23 WO disclosed