SCHEMBL16623504

SCHEMBL16623504

N=C(c1csc(C(N)=O)c1)c1c(Nc2ccccn2)cc[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.43
NPC1 O15118 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TP53 P04637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
JAK2 O60674 5/20 0.36
JAK3 P52333 3/20 0.36
NTRK1 P04629 2/20 0.35
JAK1 P23458 4/20 0.34
TYK2 P29597 4/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPK10 P53779 1/20 0.33
GFER P55789 1/20 0.33
MAPT P10636 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16726647 0.80
SCHEMBL16726667 0.78 HPGD (0.31) MEN1KMT2AHTT
SCHEMBL16726671 0.75 HPGD (0.34) HTT
SCHEMBL16623551 0.75 JAK1 (0.34) JAK2JAK3JAK1TYK2
SCHEMBL16623491 0.74 JAK1 (0.34) JAK2JAK1TYK2
SCHEMBL17849195 0.74 HSP90AA1 (0.35) JAK2JAK3JAK1TYK2
SCHEMBL16623536 0.74 HSP90AA1 (0.35) JAK2JAK3JAK1TYK2
SCHEMBL16623474 0.74 HSP90AA1 (0.35) JAK2JAK3JAK1TYK2
SCHEMBL16623510 0.74 JAK1 (0.42) JAK2JAK3JAK1TYK2
SCHEMBL16623472 0.74 JAK1 (0.33) JAK2JAK3JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed