SCHEMBL16623527

SCHEMBL16623527

N=C(c1ccc(OF)cc1)c1c(NC2CCCC2)cc[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 9/20 0.36
JAK2 O60674 6/20 0.36
BRD4 O60885 1/20 0.35
ROCK1 Q13464 1/20 0.32
HCAR3 P49019 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
MAPK1 P28482 1/20 0.31
F2 P00734 1/20 0.31
PLG P00747 1/20 0.31
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
PRSS3 P35030 1/20 0.31
ST14 Q9Y5Y6 1/20 0.31
ALOX15 P16050 1/20 0.31
EPHX2 P34913 2/20 0.31
KDM4E B2RXH2 1/20 0.31
NUAK1 O60285 1/20 0.30
PDGFRA P16234 1/20 0.30
TYK2 P29597 1/20 0.30
FLT3 P36888 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16726649 0.88 EPHX2 (0.41) JAK1JAK2BRD4EPHX2
SCHEMBL16726651 0.87 NPC1 (0.41) JAK1JAK2BRD4EPHX2KDM4E
SCHEMBL16623555 0.86 JAK1 (0.38) JAK1JAK2BRD4HCAR3HDAC8
SCHEMBL16623464 0.85 JAK1 (0.38) JAK1JAK2BRD4HCAR3HDAC8
SCHEMBL16623528 0.85 RAB9A (0.41) JAK1JAK2BRD4HDAC8ALOX15
SCHEMBL16623521 0.84 JAK1 (0.39) JAK1JAK2KDM4ENUAK1PDGFRA
SCHEMBL16623515 0.84 PARP1 (0.41) JAK1JAK2EPHX2
SCHEMBL16623542 0.84 JAK1 (0.39) JAK1JAK2BRD4HCAR3HDAC8
SCHEMBL16623524 0.84 JAK1 (0.37) JAK1JAK2BRD4HCAR3HDAC8
SCHEMBL16623525 0.83 JAK1 (0.36) JAK1JAK2BRD4HCAR3HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857400-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-04-08 EP disclosed