SCHEMBL16624727

SCHEMBL16624727

C=C/C(=C\C)C(OCc1ccc2c(c1)OCc1cc(COCc3cccc(C(=O)OC)c3)ccc1-2)(c1ccc(OC)cc1)c1ccc(OC)cc1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 18/20 0.43
ROCK1 Q13464 1/20 0.38
MRGPRX4 Q96LA9 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624717 0.89 ROCK2 (0.35) ROCK2ROCK1
SCHEMBL16627087 0.86 ROCK2 (0.35) ROCK2ROCK1
SCHEMBL16624702 0.85 ROCK2 (0.46) ROCK2ROCK1MRGPRX4
SCHEMBL16624715 0.78 ROCK2 (0.46) ROCK2ROCK1MRGPRX4
SCHEMBL18165313 0.76 SMPD1 (0.43) ROCK2ROCK1MRGPRX4
SCHEMBL16624706 0.76 ROCK2 (0.48) ROCK2ROCK1
SCHEMBL22540469 0.76 ROCK2 (0.35) ROCK2ROCK1
SCHEMBL16624701 0.72 ROCK2 (0.38) ROCK2ROCK1
SCHEMBL16624806 0.71 ROCK2 (0.38) ROCK2ROCK1
SCHEMBL16624700 0.68 ROCK2 (0.41) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050871-A2 ORGANIC COMPOUNDS TO TREAT HEPATITIS B VIRUS NOVARTIS AG (CH) 2015-04-09 WO disclosed
WO-2015051366-A2 NOVEL FORMATS FOR ORGANIC COMPOUNDS FOR USE IN RNA INTERFERENCE NOVARTIS AG (CH) 2015-04-09 WO disclosed