SCHEMBL16625847

SCHEMBL16625847

O=C(c1ccc(-c2ccc3ncc(-c4ccnc5[nH]ccc45)n3n2)cc1)N1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 15/20 0.61
MKNK2 Q9HBH9 15/20 0.61
EIF4E P06730 5/20 0.56
CHEK1 O14757 1/20 0.50
PIK3CA P42336 1/20 0.50
ATR Q13535 1/20 0.50
CYP3A4 P08684 1/20 0.50
PRKCA P17252 1/20 0.47
PRKCI P41743 1/20 0.47
PRKCE Q02156 1/20 0.47
TAF1 P21675 1/20 0.46
LRRK2 Q5S007 1/20 0.45
FYN P06241 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16626044 0.90 MKNK1 (0.62) MKNK1MKNK2EIF4ECHEK1PIK3CA
SCHEMBL16620611 0.85 MKNK1 (0.53) MKNK1MKNK2EIF4ECHEK1PIK3CA
SCHEMBL4873430 0.84 IKBKB (0.60) PIK3CACYP3A4PRKCITAF1LRRK2
SCHEMBL16304077 0.79 MKNK1 (0.78) MKNK1MKNK2EIF4ECYP3A4FYN
SCHEMBL17998738 0.79 MKNK1 (0.52) MKNK1MKNK2EIF4ECYP3A4TAF1
SCHEMBL16621060 0.77 MKNK1 (0.50) MKNK1MKNK2EIF4ECYP3A4TAF1
SCHEMBL22689133 0.77 MKNK1 (0.68) MKNK1MKNK2EIF4ECYP3A4
SCHEMBL16620475 0.77 MKNK1 (0.68) MKNK1MKNK2EIF4ECYP3A4
SCHEMBL16626028 0.76 MKNK1 (0.53) MKNK1MKNK2EIF4ECYP3A4
SCHEMBL29756282 0.76 MKNK1 (0.51) MKNK1MKNK2EIF4ECYP3A4TAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050505-A1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2015-04-09 WO disclosed