SCHEMBL16628707

SCHEMBL16628707

CCCc1ccc2nc(N)nc(C(=O)N(CC)CC)c2c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
DHFR P00374 1/20 0.38
HSP90AA1 P07900 2/20 0.37
ASIC3 Q9UHC3 1/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3092345 0.90 ALDH1A1 (0.41) ALDH1A1HPGDLMNADHFR
SCHEMBL3088463 0.83 HSP90AA1 (0.53) ALDH1A1HPGDLMNADHFRHSP90AA1
SCHEMBL13144829 0.82 ALDH1A1 (0.41) ALDH1A1HPGDLMNADHFRHSP90AA1
SCHEMBL3088521 0.82 HSP90AB1 (0.45) ALDH1A1HPGDLMNA
SCHEMBL3087968 0.82 HSP90AA1 (0.47) ALDH1A1HPGDLMNADHFRHSP90AA1
SCHEMBL3089581 0.80 HPGD (0.50) ALDH1A1HPGDLMNADHFRHSP90AA1
SCHEMBL3097002 0.80 HSP90AA1 (0.48) ALDH1A1HPGDLMNADHFRHSP90AA1
SCHEMBL16628739 0.80 IP6K1 (0.44) ALDH1A1HPGDLMNADHFRHSP90AA1
SCHEMBL3099114 0.79 HSP90AA1 (0.49) ALDH1A1DHFRHSP90AA1
SCHEMBL3099210 0.79 ADORA3 (0.54) ALDH1A1HPGDLMNAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP claimed
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP disclosed