SCHEMBL16628733

SCHEMBL16628733

Cc1cccc(CCNC(=O)c2nc(N)nc3ccccc23)c1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.59
ADORA1 P30542 4/20 0.59
RAB9A P51151 3/20 0.57
NPC1 O15118 2/20 0.57
ADORA3 P0DMS8 3/20 0.56
APP P05067 1/20 0.55
ADORA2B P29275 1/20 0.51
MAPT P10636 3/20 0.50
RXFP1 Q9HBX9 2/20 0.50
LMNA P02545 2/20 0.49
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
POLB P06746 1/20 0.48
TP53 P04637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3081056 0.88 ADORA2A (0.70) ADORA2AADORA1RAB9ANPC1ADORA3
SCHEMBL16628795 0.87 ADORA3 (0.66) ADORA2AADORA1RAB9ANPC1ADORA3
SCHEMBL3090422 0.86 ADORA2A (0.65) ADORA2AADORA1RAB9ANPC1ADORA3
SCHEMBL16628794 0.86 ADORA3 (0.58) ADORA2AADORA1RAB9ANPC1ADORA3
SCHEMBL16628768 0.84 ADORA2A (0.54) ADORA2AADORA1ADORA3ADORA2BMAPT
SCHEMBL16628738 0.84 ADORA2A (0.59) ADORA2AADORA1ADORA3APPADORA2B
SCHEMBL3093862 0.82 ADORA2A (0.62) ADORA2AADORA1RAB9ANPC1ADORA3
SCHEMBL16628808 0.81 ADORA2A (0.55) ADORA2AADORA1RAB9AADORA3ADORA2B
SCHEMBL3075309 0.81 NPC1 (0.56) ADORA2AADORA1RAB9ANPC1ADORA3
SCHEMBL16628774 0.81 RAB9A (0.58) ADORA2AADORA1RAB9ANPC1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP claimed