SCHEMBL16628741

SCHEMBL16628741

CN(C)CCCNC(=O)c1nc(N)nc2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.61
ADORA3 P0DMS8 5/20 0.55
ADORA2A P29274 2/20 0.51
ADORA1 P30542 2/20 0.51
ADORA2B P29275 1/20 0.51
KMT2A Q03164 2/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
SLC2A1 P11166 1/20 0.50
APOBEC3A P31941 1/20 0.50
RAD52 P43351 1/20 0.50
RAB9A P51151 1/20 0.50
APOBEC3G Q9HC16 1/20 0.50
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ALOX15 P16050 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3096053 0.86 ADORA3 (0.59) HTTADORA3ADORA2AADORA1ADORA2B
SCHEMBL16628837 0.85 ADORA3 (0.58) ADORA3ADORA2AADORA1ADORA2BKMT2A
SCHEMBL3094118 0.85 ADORA3 (0.58) HTTADORA3ADORA2AADORA1ADORA2B
SCHEMBL3087918 0.83 ADORA3 (0.62) ADORA3ADORA2AADORA1ADORA2BNPC1
SCHEMBL3085053 0.83 ADORA3 (0.55) HTTADORA3ADORA2AADORA1ADORA2B
SCHEMBL3093862 0.82 ADORA2A (0.62) ADORA3ADORA2AADORA1ADORA2BNPC1
SCHEMBL3081056 0.81 ADORA2A (0.70) ADORA3ADORA2AADORA1ADORA2BNPC1
SCHEMBL3093664 0.81 ADORA3 (0.55) ADORA3ADORA2AADORA1ADORA2BKMT2A
SCHEMBL3087861 0.80 ADORA3 (0.65) HTTADORA3ADORA2AADORA1ADORA2B
SCHEMBL3081770 0.80 ADORA3 (0.58) HTTADORA3ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP claimed