SCHEMBL16628744

SCHEMBL16628744

Nc1nc(C(=O)NCCc2ccccn2)c2ccccc2n1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.71
ADORA1 P30542 4/20 0.71
ADORA3 P0DMS8 4/20 0.58
ADORA2B P29275 1/20 0.58
SMN1; SMN2 Q16637 3/20 0.55
KDM4E B2RXH2 2/20 0.55
HPGD P15428 1/20 0.54
RAB9A P51151 4/20 0.52
NPC1 O15118 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
LMNA P02545 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP3A4 P08684 1/20 0.48
PTGFR P43088 1/20 0.48
NAMPT P43490 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3081056 0.85 ADORA2A (0.70) ADORA2AADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL16628774 0.80 RAB9A (0.58) ADORA2AADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL3087918 0.80 ADORA3 (0.62) ADORA2AADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL3087954 0.80 ADORA2A (0.66) ADORA2AADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL16628795 0.80 ADORA3 (0.66) ADORA2AADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL3093862 0.79 ADORA2A (0.62) ADORA2AADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL3089577 0.79 ADORA2A (0.65) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL16628808 0.79 ADORA2A (0.55) ADORA2AADORA1ADORA3ADORA2BHPGD
SCHEMBL3096049 0.78 ADORA2A (0.55) ADORA2AADORA1ADORA3ADORA2BSMN1; SMN2
SCHEMBL483578 0.78 RAB9A (0.74) SMN1; SMN2RAB9ANPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP claimed