SCHEMBL16628751

SCHEMBL16628751

COc1ccccc1CCNC(=O)c1nc(N)nc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.56
APBA1 Q02410 1/20 0.56
ADORA3 P0DMS8 3/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
MAPT P10636 1/20 0.54
ADORA2A P29274 9/20 0.53
MTNR1A P48039 1/20 0.53
MTNR1B P49286 1/20 0.53
ADORA1 P30542 3/20 0.53
ADORA2B P29275 1/20 0.53
POLB P06746 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HPGD P15428 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3086944 0.88 ADORA3 (0.49) CACNA1BAPBA1ADORA3MEN1KMT2A
SCHEMBL16628808 0.85 ADORA2A (0.55) ADORA3MAPTADORA2AADORA1ADORA2B
SCHEMBL16628820 0.83 ADORA3 (0.68) CACNA1BAPBA1ADORA3MEN1KMT2A
SCHEMBL3089577 0.83 ADORA2A (0.65) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL3081056 0.82 ADORA2A (0.70) ADORA3MAPTADORA2AADORA1ADORA2B
SCHEMBL16628837 0.81 ADORA3 (0.58) ADORA3MEN1KMT2AMAPTADORA2A
SCHEMBL16628794 0.81 ADORA3 (0.58) ADORA3KMT2AMAPTADORA2AADORA1
SCHEMBL3087918 0.80 ADORA3 (0.62) ADORA3ADORA2AADORA1ADORA2BHPGD
SCHEMBL16628795 0.79 ADORA3 (0.66) ADORA3MEN1KMT2AMAPTADORA2A
SCHEMBL3087954 0.79 ADORA2A (0.66) ADORA3ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164833-B1 Quinazolinamide derivatives useful for the treatment of tumour diseases MERCK PATENT GMBH (DE) 2015-04-15 EP claimed