SCHEMBL16629034

SCHEMBL16629034

CC(C)(C)c1nc(CCNCl)no1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.32
EPHA2 P29317 1/20 0.31
EPHB4 P54760 1/20 0.31
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188155 0.84 HDAC4 (0.31) CXCR3
Hydrochloric Acid SCHEMBL3707118 0.82 CNR2 (0.30) CNR2
SCHEMBL10058001 0.77 ALDH1A1 (0.42) CXCR3EPHA2EPHB4CNR2
SCHEMBL2831415 0.76 AOC3 (0.35) CXCR3
SCHEMBL21325031 0.76 CXCR3 (0.31) CXCR3
SCHEMBL4398054 0.76 PIK3CG (0.35) CXCR3
SCHEMBL22544835 0.76 CXCR3 (0.31) CXCR3EPHA2EPHB4
SCHEMBL21690696 0.76 CXCR3 (0.31) CXCR3
SCHEMBL478959 0.75 CNR2 (0.33) CXCR3EPHA2EPHB4CNR2
Hydrochloric Acid SCHEMBL3712851 0.74 AOC3 (0.35) CXCR3CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9751888-B2 Heterocyclic compounds and uses thereof INFINITY PHARMACEUTICALS, INC. (US) 2017-09-05 US disclosed
US-20160222016-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF TWELVE THERAPEUTICS, INC. 2016-08-04 US disclosed
WO-2015051241-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF INFINITY PHARMACEUTICALS, INC. (US) 2015-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160222016-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PIK3CA, PIK3CD, PIK3CB CXCR3 1282/4885EPHA2 1751/4885EPHB4 3502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.