SCHEMBL16629839

SCHEMBL16629839

CC(c1cnccn1)N(C)C(=O)c1ccc(C[C@@H]2CC[C@H](Cc3ccc(Cl)nc3)N2)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
ADRB3 P13945 2/20 0.33
KMT2A Q03164 4/20 0.33
MEN1 O00255 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
EPHX1 P07099 1/20 0.32
LMNA P02545 1/20 0.32
SLC6A4 P31645 1/20 0.32
MDM2 Q00987 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16619499 0.88 ADRB3 (0.44) ADRB3SLC6A4
SCHEMBL16619700 0.88 ADRB3 (0.44) ADRB3SLC6A4
SCHEMBL16619680 0.81 ADRB3 (0.50) ADRB3SLC6A4
SCHEMBL16619677 0.79 ADRB3 (0.43) ADRB3SLC6A4
SCHEMBL16618866 0.76 ADRB3 (0.53) ADRB3KMT2AMEN1ALDH1A1MAPT
SCHEMBL16618864 0.76 ADRB3 (0.53) ADRB3KMT2AMEN1ALDH1A1MAPT
SCHEMBL16629885 0.75 LMNA (0.43) LMNA
SCHEMBL18210816 0.73 IDO1 (0.37) ADRB3KMT2AMEN1NPC1RAB9A
SCHEMBL21278187 0.73 ADRB3 (0.43) ADRB3
SCHEMBL16630638 0.72 PSEN1 (0.39) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015050798-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2015-04-09 WO disclosed