SCHEMBL16632699

SCHEMBL16632699

N#Cc1cc2c(Br)cc(Cl)cc2o1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.50
CYP2A6 P11509 1/20 0.38
PSMB8 P28062 2/20 0.33
PSMB5 P28074 1/20 0.33
AHR P35869 2/20 0.31
F2RL3 Q96RI0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16632656 0.79 CYP2A6 (0.38) CYP2A6F2RL3
SCHEMBL16632564 0.75 MCL1 (0.58) MCL1AHRF2RL3
SCHEMBL16632353 0.73 CYP2A6 (0.52) CYP2A6PSMB8F2RL3
SCHEMBL16345161 0.72 MCL1 (0.54) MCL1AHR
SCHEMBL16345100 0.69 MCL1 (0.51) MCL1AHR
SCHEMBL18325887 0.68 MCL1 (0.50) MCL1AHR
SCHEMBL16345420 0.68 MCL1 (0.54) MCL1AHR
SCHEMBL28730094 0.68 MCL1 (0.50) MCL1AHR
SCHEMBL16632531 0.67 SLC6A4 (0.42) CYP2A6
SCHEMBL6779123 0.66 MCL1 (0.51) MCL1CYP2A6AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382245-B2 Compounds and methods for treating HIV infections YALE UNIVERSITY (US) 2016-07-05 US disclosed
US-20150105351-A1 COMPOUNDS AND METHODS FOR TREATING HIV INFECTIONS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150105351-A1 COMPOUNDS AND METHODS FOR TREATING HIV INFECTIONS POLM, POLRMT, DHFR MCL1 2386/4885CYP2A6 785/4885PSMB8 3011/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.