SCHEMBL16634636

SCHEMBL16634636

O=C(O)c1ccc(-n2c(=O)n(C(=O)c3c(Cl)cccc3C(F)(F)F)c3ccccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RORC P51449 18/20 0.56
CYP3A4 P08684 3/20 0.56
CYP2C9 P11712 3/20 0.56
PPARG P37231 2/20 0.56
CYP2C19 P33261 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634554 0.89 RORC (0.55) RORCCYP3A4CYP2C9CYP2C19
SCHEMBL16634596 0.85 RORC (0.61) RORCCYP3A4CYP2C9PPARGCYP2C19
SCHEMBL16634653 0.84 RORC (0.60) RORCCYP3A4CYP2C9PPARGCYP2C19
SCHEMBL16634706 0.81 RORC (0.48) RORCCYP3A4CYP2C9PPARGCYP2C19
SCHEMBL16634830 0.78 RORC (0.43) RORCCYP3A4CYP2C9CYP2C19
SCHEMBL16634779 0.78 RORC (0.53) RORCCYP3A4CYP2C9PPARGCYP2C19
SCHEMBL16634652 0.77 RORC (0.50) RORCCYP3A4CYP2C9PPARGCYP2C19
SCHEMBL16634775 0.77 RORC (0.63) RORCCYP3A4CYP2C9PPARGCYP2C19
SCHEMBL16634618 0.76 RORC (0.45) RORCCYP3A4CYP2C9PPARGCYP2C19
SCHEMBL16634647 0.76 RORC (0.54) RORCCYP3A4CYP2C9PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed