SCHEMBL16635078

SCHEMBL16635078

O=C(NCc1cncc(Br)c1)C1CC(F)CN1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CFD P00746 14/20 0.48
TRPA1 O75762 5/20 0.47
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16635165 1.00 CFD (0.48) CFDTRPA1SMN1; SMN2
SCHEMBL16648088 0.85 FNTA (0.46) CFDTRPA1
SCHEMBL16635467 0.83 TRPA1 (0.46) CFDTRPA1
SCHEMBL16635520 0.79 TRPA1 (0.47) CFDTRPA1
SCHEMBL16635433 0.79 TRPA1 (0.73) TRPA1
SCHEMBL18546533 0.78 CFD (0.60) CFD
SCHEMBL16635248 0.78 TRPA1 (0.47) CFDTRPA1
SCHEMBL16635061 0.78 TRPA1 (0.49) CFDTRPA1
SCHEMBL17959669 0.76 TRPA1 (0.47) CFDTRPA1
SCHEMBL16634887 0.76 TRPA1 (0.47) CFDTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3055302-A1 SUBSTITUTED HETEROCYCLIC SULFONAMIDE COMPOUNDS USEFUL AS TRPA1 MODULATORS F. Hoffmann-La Roche AG (CH) 2016-08-17 EP disclosed
WO-2015052264-A1 SUBSTITUTED HETEROCYCLIC SULFONAMIDE COMPOUNDS USEFUL AS TRPA1 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2015-04-16 WO disclosed