SCHEMBL16635641

SCHEMBL16635641

CC1(F)CC(C(=O)NCc2cc(F)cc(Br)c2)N(C(=O)O)C1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.46
CFD P00746 14/20 0.38
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16635012 0.89 TRPA1 (0.39) TRPA1CFDALDH1A1
SCHEMBL17959577 0.86 TRPA1 (0.44) TRPA1CFDALDH1A1
SCHEMBL16647938 0.86 TRPA1 (0.44) TRPA1CFDALDH1A1
SCHEMBL16634985 0.79 TRPA1 (0.71) TRPA1
SCHEMBL16647810 0.79 TRPA1 (0.71) TRPA1
SCHEMBL16635044 0.79 TRPA1 (0.71) TRPA1
SCHEMBL16634840 0.79 ALDH1A1 (0.39) TRPA1ALDH1A1
SCHEMBL16635467 0.77 TRPA1 (0.46) TRPA1CFD
SCHEMBL16647936 0.76 HDAC8 (0.39) TRPA1CFDALDH1A1
SCHEMBL17959575 0.76 HDAC8 (0.39) TRPA1CFDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3055302-A1 SUBSTITUTED HETEROCYCLIC SULFONAMIDE COMPOUNDS USEFUL AS TRPA1 MODULATORS F. Hoffmann-La Roche AG (CH) 2016-08-17 EP disclosed
WO-2015052264-A1 SUBSTITUTED HETEROCYCLIC SULFONAMIDE COMPOUNDS USEFUL AS TRPA1 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2015-04-16 WO disclosed