SCHEMBL1663652

SCHEMBL1663652

Nc1ccc(-c2n[nH]c3ccc(O)cc23)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 2/20 0.68
FGFR2 P21802 2/20 0.68
MAP2K4 P45985 7/20 0.62
MAPK1 P28482 5/20 0.62
MAPKAPK3 Q16644 5/20 0.62
MAPK6 Q16659 5/20 0.62
MAPKAPK2 P49137 3/20 0.62
MAPKAPK5 Q8IW41 2/20 0.62
PDPK1 O15530 1/20 0.60
HSP90AB1 P08238 1/20 0.60
FGFR3 P22607 1/20 0.54
AXL P30530 2/20 0.48
MKNK1 Q9BUB5 1/20 0.46
JAK2 O60674 3/20 0.45
DCLK1 O15075 1/20 0.45
PRKD3 O94806 1/20 0.45
MAP4K4 O95819 1/20 0.45
CHEK2 O96017 1/20 0.45
CSF1R P07333 1/20 0.45
FER P16591 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663211 0.86 AXL (0.60) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL14359839 0.83 MAP2K4 (0.62) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL5378056 0.83 DCLK1 (0.65) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL10130802 0.78 JAK2 (0.60) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
Hydrochloric Acid SCHEMBL10369298 0.77 JAK2 (0.58) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL4006856 0.77 AXL (0.55) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL2469031 0.77 AXL (0.55) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL22801614 0.77 MAP2K4 (1.00) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL4029036 0.77 MAP2K4 (0.67) FGFR1FGFR2MAP2K4MAPK1MAPKAPK3
SCHEMBL12193658 0.76 MKNK1 (0.61) FGFR1FGFR2MAPK1PDPK1AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2642994-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS Ligand Pharmaceuticals Incorporated (US) 2013-10-02 EP disclosed
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2012068406-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS LIGAND PHARMACEUTICALS INCORPORATED (US) 2012-05-24 WO disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed