SCHEMBL16637129

SCHEMBL16637129

Cc1nn(-c2nccs2)cc1-c1ccc(NC(=O)c2ccc(F)c(F)c2F)cc1F

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 4/20 0.36
ADORA2A P29274 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
IDO1 P14902 2/20 0.35
DNM1L O00429 1/20 0.35
AVPR2 P30518 1/20 0.34
GPR27 Q9NS67 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
S1PR1 P21453 1/20 0.34
BTK Q06187 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23833354 0.90 ALDH1A1 (0.35) NR3C1ADORA2ACYP3A4CYP2C19NPC1
SCHEMBL16636671 0.90 MEN1 (0.37) NR3C1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL16636788 0.88 MEN1 (0.44) ADORA2ACYP3A4CYP2C19NPC1RAB9A
SCHEMBL16637313 0.85 TP53 (0.42) NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL16636848 0.85 MGAM (0.37) NPC1RAB9ASMN1; SMN2KDM4ES1PR1
SCHEMBL18038398 0.84 BUB1 (0.39) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL16636702 0.84 MAOB (0.38) ADORA2ACYP3A4CYP2C19NPC1RAB9A
SCHEMBL29420780 0.84 BUB1 (0.39) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL16637004 0.83 IL2 (0.39) ADORA2ACYP3A4CYP2C19NPC1RAB9A
SCHEMBL16636521 0.82 NPC1 (0.45) ADORA2ACYP3A4CYP2C19NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9611263-B2 Compounds that modulate intracellular calcium CALCIMEDICA, INC. (US) 2017-04-04 US disclosed
US-20160229845-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM AVENUE CAPITAL MANAGEMENT II, L.P. 2016-08-11 US disclosed
WO-2015054283-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2015-04-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160229845-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM ORAI1, SARAF, RYR2 NR3C1 4202/4885ADORA2A 1775/4885CYP3A4 4329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.