SCHEMBL16637467

SCHEMBL16637467

CC(CF)Cc1ccc(C(C)C(=O)O)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.69
PTGS1 P23219 12/20 0.69
AKR1C3 P42330 3/20 0.69
LMNA P02545 2/20 0.69
CYP2C9 P11712 2/20 0.69
CXCR1 P25024 2/20 0.69
CXCR2 P25025 2/20 0.69
AKR1C2 P52895 2/20 0.69
ALB P02768 1/20 0.69
ESR1 P03372 1/20 0.69
ALOX5 P09917 1/20 0.69
RARB P10826 1/20 0.69
ADRB3 P13945 1/20 0.69
NFKB1 P19838 1/20 0.69
HTR2A P28223 1/20 0.69
NR1I3 Q14994 1/20 0.69
SLC22A6 Q4U2R8 1/20 0.69
CXCL8 P10145 1/20 0.69
TSHR P16473 1/20 0.69
BLM P54132 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24209440 0.84 PTGS2 (0.71) PTGS2PTGS1AKR1C3LMNACYP2C9
SCHEMBL16943972 0.84 PTGS2 (0.71) PTGS2PTGS1AKR1C3LMNACYP2C9
SCHEMBL31389025 0.84 PTGS2 (0.71) PTGS2PTGS1AKR1C3LMNACYP2C9
Ibuprofen SCHEMBL3001 0.82 PTGS1 (1.00) PTGS2PTGS1AKR1C3LMNACYP2C9
SCHEMBL7622372 0.82 PTGS2 (0.67) PTGS2PTGS1AKR1C3LMNACYP2C9
Ibuprofen SCHEMBL8754799 0.82 PTGS1 (1.00) PTGS2PTGS1AKR1C3LMNACYP2C9
Ibuprofen SCHEMBL19439560 0.82 PTGS1 (1.00) PTGS2PTGS1AKR1C3LMNACYP2C9
Ibuprofen SCHEMBL239446 0.82 PTGS1 (1.00) PTGS2PTGS1AKR1C3LMNACYP2C9
Ibuprofen SCHEMBL19439559 0.82 PTGS1 (1.00) PTGS2PTGS1AKR1C3LMNACYP2C9
Dexibuprofen SCHEMBL30091137 0.82 PTGS1 (1.00) PTGS2PTGS1AKR1C3LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015134467-A1 METHODS AND COMPOSITIONS FOR DIRECT RADIOACTIVE LABELING OF BIO-ACTIVE MOLECULES AND BUILDING BLOCKS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2015-09-11 WO disclosed
WO-2015054476-A1 C-HALOGEN BOND FORMATION THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2015-04-16 WO disclosed