SCHEMBL16637637

SCHEMBL16637637

CCc1nn(-c2nccs2)cc1-c1ccc(N(C(=O)c2ccccc2F)c2ccccc2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
S1PR1 P21453 5/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
CASP3 P42574 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
ALDH1A1 P00352 2/20 0.31
PPARG P37231 1/20 0.31
NCOA2 Q15596 1/20 0.31
NCOA1 Q15788 1/20 0.31
S1PR3 Q99500 2/20 0.30
S1PR4 O95977 1/20 0.30
S1PR5 Q9H228 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
RAB9A P51151 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16644206 0.81 KDM4E (0.33) KDM4EKMT2ALMNA
SCHEMBL16636877 0.80 SMN1; SMN2 (0.38) KDM4EMEN1KMT2ARAB9ALMNA
SCHEMBL16636486 0.76 IL2 (0.37) KDM4EALDH1A1MEN1KMT2AHTT
SCHEMBL16636755 0.74 IL2 (0.45) KDM4EALDH1A1MEN1KMT2AHTT
SCHEMBL16636856 0.74 MAPT (0.45) KDM4EALDH1A1MEN1KMT2ARAB9A
SCHEMBL17997393 0.71 CYP1A2 (0.38) KDM4ECYP1A2ALDH1A1PPARGNCOA2
SCHEMBL17997392 0.69 KMT2A (0.34) KDM4EKMT2ALMNA
SCHEMBL16636669 0.69 POLB (0.41) KDM4EALDH1A1MEN1KMT2ARAB9A
SCHEMBL31222089 0.68 L3MBTL1 (0.47) KDM4EALDH1A1MEN1KMT2ARAB9A
SCHEMBL16636716 0.67 IL2 (0.45) MEN1KMT2ARAB9ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015054283-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2015-04-16 WO disclosed