SCHEMBL16637829

SCHEMBL16637829

COC(=O)[C@@H]1CCCC[C@H]1c1nc(Oc2ccccc2)sc1-c1ccc(N2CCSC(O)(O)C2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.40
SLC6A4 P31645 3/20 0.40
CPT2 P23786 1/20 0.38
CPT1A P50416 1/20 0.38
CTSK P43235 2/20 0.36
ALDH1A1 P00352 6/20 0.33
USP2 O75604 6/20 0.33
HSD17B10 Q99714 6/20 0.33
CYP3A4 P08684 5/20 0.33
CYP1A2 P05177 4/20 0.33
CYP2C9 P11712 4/20 0.33
HIF1A Q16665 3/20 0.33
MAPK1 P28482 2/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 2/20 0.32
GAA P10253 1/20 0.32
SCN9A Q15858 1/20 0.32
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
SMN1; SMN2 Q16637 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637539 0.92 CTSK (0.36) CTSKALDH1A1USP2HSD17B10CYP3A4
SCHEMBL16636094 0.84 SLC6A2 (0.42) SLC6A2SLC6A4CPT2CPT1ACTSK
SCHEMBL16636575 0.84 CTSK (0.49) SLC6A2SLC6A4CPT2CPT1ACTSK
SCHEMBL16636097 0.84 CTSK (0.49) SLC6A2SLC6A4CPT2CPT1ACTSK
SCHEMBL16637719 0.76 CTSK (0.39) SLC6A2SLC6A4CTSKALDH1A1KMT2A
SCHEMBL16636142 0.75 CTSK (0.49) CTSKALDH1A1BTK
SCHEMBL16635864 0.75 CTSK (0.49) CTSKALDH1A1BTK
SCHEMBL16636141 0.75 CTSK (0.42) CTSKALDH1A1TSHRKMT2ABTK
SCHEMBL16635863 0.75 CTSK (0.42) CTSKALDH1A1TSHRKMT2ABTK
SCHEMBL16635949 0.73 SLC6A2 (0.48) SLC6A2SLC6A4CPT2CPT1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051479-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-04-16 WO disclosed