SCHEMBL16637898

SCHEMBL16637898

N=S1(=O)CCN(c2ccc(Br)cc2)CC1.O=C(N=S1(=O)CCN(c2ccc(Br)cc2)CC1)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 4/20 0.35
KMT2A Q03164 2/20 0.34
USP2 O75604 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
ALDH1A1 P00352 2/20 0.33
ABHD6 Q9BV23 1/20 0.33
CCR1 P32246 1/20 0.33
F10 P00742 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
MEN1 O00255 1/20 0.32
APAF1 O14727 1/20 0.32
MAPK1 P28482 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
EIF4H Q15056 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16635667 0.94 AKR1C3 (0.40) AKR1C3KDM4EMAPTKMT2AUSP2
SCHEMBL16635950 0.80 AKR1C3 (0.44) AKR1C3KDM4EMAPTKMT2AUSP2
SCHEMBL16793360 0.73 PANK3 (0.38) ALDH1A1
SCHEMBL16635687 0.72 F11 (0.44) KDM4EALDH1A1ABHD6F10SMN1; SMN2
SCHEMBL16635824 0.71 AKR1C3 (0.41) AKR1C3KDM4EMAPTKMT2AUSP2
SCHEMBL16635670 0.68 AKR1C3 (0.40) AKR1C3MAPTKMT2AUSP2DRD2
SCHEMBL1235260 0.67 KDM4E (0.59) AKR1C3KDM4EMAPTKMT2AUSP2
SCHEMBL20639966 0.66 AKR1C3 (0.58) AKR1C3MAPTKMT2AUSP2ALDH1A1
SCHEMBL20640032 0.66 MLYCD (0.50) AKR1C3KDM4EMAPTKMT2AUSP2
SCHEMBL23624939 0.64 MAPT (0.55) KDM4EMAPTKMT2AUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015051479-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-04-16 WO disclosed