SCHEMBL16638752

SCHEMBL16638752

Cc1ccc(-c2ccc(-c3ccc(C4CCC(I)CC4)cc3)c(F)c2F)cc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.39
AKR1C3 P42330 3/20 0.37
AKR1C2 P52895 3/20 0.37
AKR1B10 O60218 2/20 0.37
AKR1C4 P17516 2/20 0.37
AKR1C1 Q04828 2/20 0.37
CYP3A4 P08684 3/20 0.37
CYP2C9 P11712 2/20 0.37
APP P05067 2/20 0.37
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
NISCH Q9Y2I1 1/20 0.34
KDM1A O60341 1/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
PRKAB2 O43741 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA2 P54646 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL803146 0.88 ESR2 (0.41) SLC6A3AKR1C3AKR1C2AKR1B10AKR1C4
SCHEMBL26167206 0.81 CYP3A4 (0.38) SLC6A3CYP3A4CYP2C9APPCYP2D6
SCHEMBL4549771 0.80 CYP3A4 (0.41) SLC6A3AKR1C3AKR1C2AKR1B10AKR1C4
SCHEMBL10037540 0.77 ESR2 (0.36) CYP3A4CYP2C9APPCYP2D6CYP2C19
SCHEMBL18069652 0.77 AKR1C3 (0.50) AKR1C3AKR1C2AKR1B10AKR1C4AKR1C1
SCHEMBL12075617 0.77 CYP3A4 (0.39) SLC6A3AKR1C3AKR1C2AKR1B10AKR1C4
SCHEMBL26672922 0.77 CYP3A4 (0.36) SLC6A3CYP3A4CYP2C9APPCYP2D6
SCHEMBL18736336 0.77 SLC6A3 (0.36) SLC6A3
SCHEMBL24661359 0.77 AKR1C3 (0.43) SLC6A3AKR1C3AKR1C2AKR1B10AKR1C4
SCHEMBL12056677 0.76 NPC1 (0.37) CYP3A4CYP2C9APPCYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9005720-B2 Liquid-crystal display MERCK PATENT GMBH (DE) 2015-04-14 US disclosed