SCHEMBL16638802

SCHEMBL16638802

C=CC(C)(C)OC(=O)NNC(=O)Cc1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
GAA P10253 2/20 0.43
HTT P42858 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
SMN1; SMN2 Q16637 6/20 0.42
LMNA P02545 3/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 2/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4549800 0.85 KDM4E (0.54) KDM4EGAAHTTTDP1SMN1; SMN2
SCHEMBL4317497 0.73 HTT (0.49) KDM4EGAAHTTTDP1SMN1; SMN2
SCHEMBL1431992 0.72 ALDH1A1 (0.50) KDM4EGAAHTTSMN1; SMN2LMNA
SCHEMBL27099061 0.72 HTT (0.50) KDM4EGAAHTTTDP1SMN1; SMN2
SCHEMBL18673195 0.72 HPGD (0.54) GAAHTTSMN1; SMN2LMNAKMT2A
SCHEMBL15829741 0.71 GAA (0.50) KDM4EGAATDP1SMN1; SMN2LMNA
SCHEMBL13580096 0.71 HTT (0.49) KDM4EGAAHTTTDP1SMN1; SMN2
SCHEMBL26196694 0.71 ALDH1A1 (0.63) GAAHTTSMN1; SMN2LMNAKMT2A
SCHEMBL2068949 0.71 GAA (0.49) KDM4EGAAHTTTDP1LMNA
SCHEMBL26196749 0.71 APLNR (0.51) KDM4EGAAHTTLMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2540720-B1 1,3,4,8-TETRAHYDRO-2H-PYRIDO[1,2-A]PYRAZINE DERIVATIVE AND USE OF SAME AS HIV INTEGRASE INHIBITOR JAPAN TOBACCO INC (JP) 2015-04-15 EP disclosed