SCHEMBL16638978

SCHEMBL16638978

C=Cc1c(Cl)cccc1C1(O)CCNCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.44
DRD2 P14416 4/20 0.42
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
OPRK1 P41145 2/20 0.36
OPRL1 P41146 2/20 0.36
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
DRD3 P35462 3/20 0.32
DRD4 P21917 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
EPHB3 P54753 1/20 0.31
ADRB1 P08588 2/20 0.31
KDM1A O60341 1/20 0.31
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1513548 0.79 SIGMAR1 (0.50) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL652087 0.79 SIGMAR1 (0.57) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL2267923 0.76 SIGMAR1 (0.51) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL2270695 0.76 SIGMAR1 (0.47) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL1513275 0.75 DRD2 (0.55) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL3266597 0.73 SIGMAR1 (0.51) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL3107373 0.70 DRD2 (0.42) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL4703446 0.70 SIGMAR1 (0.48) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL8086598 0.69 SIGMAR1 (0.46) SIGMAR1DRD2OPRM1OPRD1OPRK1
SCHEMBL1660350 0.69 SIGMAR1 (0.62) SIGMAR1DRD2OPRM1HTR2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2477983-B1 (4-PHENYL-PIPERIDIN-1-YL)-[5-1H-PYRAZOL-4YL)-THIOPHEN-3-YL]-METHANONE COMPOUNDS AND THEIR USE UNIV EDINBURGH (GB) 2015-04-15 EP disclosed