SCHEMBL16638987

SCHEMBL16638987

Cc1cc(N(c2ccccc2)c2ccc(-c3ccccc3)c3ccccc23)ccc1-c1ccc2ccccc2c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.36
CYP2A6 P11509 1/20 0.36
TSHR P16473 1/20 0.36
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
ESR2 Q92731 1/20 0.33
DHFR P00374 1/20 0.33
CRHR1 P34998 1/20 0.32
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
ALDH1A1 P00352 3/20 0.31
MEN1 O00255 2/20 0.31
MAPT P10636 2/20 0.31
KMT2A Q03164 2/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16638989 0.86 CYP1A2 (0.41) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL19393502 0.84 ESR2 (0.41) CYP2A6CA12CA1CA2CA9
SCHEMBL16638997 0.84 CYP1A2 (0.42) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL16638995 0.84 CA12 (0.41) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL24514812 0.82 SIGMAR1 (0.40) CYP1A2CYP2A6CA12CA1CA2
SCHEMBL2722078 0.82 SIGMAR1 (0.42) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL29378684 0.82 SIGMAR1 (0.42) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL19292151 0.81 CA12 (0.39) CYP2A6CA12CA1CA2CA9
SCHEMBL23513194 0.80 SIGMAR1 (0.41) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL17734637 0.80 CA12 (0.45) CA12CA1CA2CA9CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2439190-B1 AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENTS TOSOH CORP (JP) 2015-04-15 EP disclosed