SCHEMBL16638989

SCHEMBL16638989

Cc1cc(N(c2ccc(-c3ccccc3)cc2)c2ccc(-c3ccccc3)cc2)ccc1-c1ccc2ccccc2c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP2A6 P11509 2/20 0.41
TSHR P16473 2/20 0.41
CA12 O43570 3/20 0.40
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA9 Q16790 3/20 0.40
ESR2 Q92731 2/20 0.34
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
PDE10A Q9Y233 1/20 0.33
MAPK1 P28482 2/20 0.32
ATM Q13315 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
CYP3A4 P08684 1/20 0.32
CASP1 P29466 1/20 0.32
RAB9A P51151 1/20 0.32
CASP7 P55210 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16638988 0.93 MAPT (0.38) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL16638995 0.92 CA12 (0.41) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL16638987 0.86 CYP1A2 (0.36) CYP1A2CYP2A6TSHRCA12CA1
SCHEMBL2604754 0.85 ESR2 (0.44) CYP1A2CYP2A6CA12CA1CA2
SCHEMBL7591957 0.85 CA12 (0.51) CA12CA1CA2CA9
SCHEMBL7596626 0.85 CA12 (0.51) CA12CA1CA2CA9
SCHEMBL16638996 0.84 CYP11B1 (0.41) CYP1A2CYP2A6TSHRALDH1A1L3MBTL1
SCHEMBL2604756 0.83 ESR2 (0.43) CYP1A2CYP2A6CA12CA1CA2
SCHEMBL2604759 0.83 ESR2 (0.43) CYP1A2CYP2A6CA12CA1CA2
SCHEMBL7596775 0.83 CA12 (0.46) CA12CA1CA2CA9ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2439190-B1 AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENTS TOSOH CORP (JP) 2015-04-15 EP disclosed