SCHEMBL1664491

SCHEMBL1664491

O=C(Nc1ccc(-n2ncc3cc(Nc4ccc(F)cc4)ccc32)cc1)c1ccc2[nH]ccc2c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
ESR1 P03372 1/20 0.47
MAPK10 P53779 4/20 0.46
MAPK8 P45983 3/20 0.46
MAOB P27338 3/20 0.46
MAOA P21397 1/20 0.46
ABL1 P00519 1/20 0.45
SMO Q99835 2/20 0.44
MAPT P10636 1/20 0.44
MAPK13 O15264 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
MAPK14 Q16539 1/20 0.43
NR3C1 P04150 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1664492 0.94 NPC1 (0.66) NPC1RAB9AESR1MAPK10MAPK8
SCHEMBL1665773 0.91 MAOB (0.56) NPC1RAB9AMAPK10MAOBMAOA
SCHEMBL1665219 0.86 MAPK10 (0.43) NPC1RAB9AMAPK10MAPK8MAOB
SCHEMBL1665249 0.84 SMO (0.54) MAPK10MAPK8MAOBSMOMAPK13
SCHEMBL1665007 0.83 MAOB (0.48) NPC1RAB9AMAOBMAOAABL1
SCHEMBL1665395 0.83 SMO (0.51) MAPK10MAPK8MAOBSMOMAPT
SCHEMBL1665429 0.83 ESR1 (0.52) NPC1RAB9AESR1MAPK10MAPK8
SCHEMBL1665083 0.82 SMO (0.52) MAPK10MAPK8MAOBSMONR3C1
SCHEMBL1665738 0.81 MAOB (0.46) NPC1RAB9AMAPK10MAOBMAOA
SCHEMBL1666769 0.81 MAOB (0.48) NPC1RAB9AMAPK10MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2642994-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS Ligand Pharmaceuticals Incorporated (US) 2013-10-02 EP disclosed
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2012068406-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS LIGAND PHARMACEUTICALS INCORPORATED (US) 2012-05-24 WO disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed